http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2022062278-A1

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filingDate 2019-12-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f87bfa1efc89aa49e16cfa944444fe20
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_157ac56127b21efe88f568183de19003
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publicationDate 2022-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2022062278-A1
titleOfInvention Small molecule inhibitors of the androgen receptor activity and/or expression and uses thereof
abstract This invention is in the field of medicinal chemistry. In particular, the invention relates to a new class of small-molecules having a piperazine (or similar) structure which function as antagonists of androgen receptor activity, and their use as therapeutics for the treatment of cancer (e.g., castration-resistant prostate cancer) and other conditions characterized with androgen receptor activity and/or androgen receptor expression.
priorityDate 2018-12-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466029722
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP51494
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465330100
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411675801
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5287969
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ29416
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415713612
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465324967
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135413511
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480871
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465967118
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465287583
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414677843
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID443460
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465961470
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416290473
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501329
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428100369
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5035
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3081349
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04838
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID82115
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451565298
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9811784
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465970318
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152566255
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP30918
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163998154
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100689318
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6058
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396839
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID241902
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID151460651
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480456
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581097
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373904
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421298036
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457797993
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422926853

Total number of triples: 1295.