http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2022041578-A1

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filingDate 2019-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_66f6b8ff9cb02420654c1767abc66736
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_67b411276a665611f9146e29542a236b
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_41a01f8278fdfeacd8c1f37fdc1c7190
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2e97a9c077cf17a5577b0f58132cb58d
publicationDate 2022-02-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2022041578-A1
titleOfInvention Isoindoline compound, and preparation method, pharmaceutical composition, and application of isoindoline compound
abstract The present invention relates to an isoindoline compound as represented by general formula (I) and used as a CRBN regulator, and a preparation method, a pharmaceutical composition, and an application of the isoindoline compound. Specifically, a class of polysubstituted isoindoline compound provided in the present invention, as a class of CRL4 CRBN E3 ubiquitin ligase regulator having a novel structure, has good anti-tumor activity and immunoregulatory activity, and can be used for preparing drugs for treating diseases associated with a CRL4 CRBN E3 ubiquitin ligase.
priorityDate 2018-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1226.