http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2021015881-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-439
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-06
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filingDate 2017-05-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b65721c6c62a2e437e051fdd235c7201
publicationDate 2021-01-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2021015881-A1
titleOfInvention Agent exhibiting antiarrhythmic effect
abstract The present invention comprises an agent exhibiting an antiarrhythmic effect, extracted from plants of genus Aconitum family Ranunculaceae, containing the alkaloids lappaconitine, N-acetylsepaconitine, 1-desmethyllappaconitine, ranaconitine, N-deacetyllappaconitine, isolappaconitine, 9-deoxy-lappaconitine or pharmaceutically acceptable salts thereof. The agent contains alkaloids in the form of hydrobromide salts of lappaconitine, N-acetylsepaconitine, 1-desmethyllappaconitine, ranaconitine, N-deacetyllappaconitine, isolappaconitine, and 9-deoxy-lappaconitine. In specific implementations, the agent may be extracted from the rhizomes and roots of the plant Aconitum septentrionale Koelle, from the rhizomes and roots of the plant Aconitum leucostomum, or from the herb of the plant Aconitum leucostomum, all of the family Ranunculaceae. A pharmaceutical composition for oral administration comprises the agent in an effective quantity and a pharmaceutically acceptable carrier. Preferably, the pharmaceutically acceptable carrier contains starch, sucrose, calcium stearate, and croscarmellose sodium. The present invention provides a more effective and safe cardioprotective agent for the prevention and treatment of arrhythmia.
priorityDate 2016-06-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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