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publicationDate 2021-01-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2021009596-A1
titleOfInvention DIARYL SUBSTITUTED 5,5-FUSED RING COMPOUNDS AS C5aR INHIBITORS
abstract The present disclosure provides, inter alia, Compounds of Formula (I) n n n n n n n n n n or pharmaceutically acceptable salts thereof that are modulators of the C5a receptor. Also provided are pharmaceutical compositions and methods of use including the treatment of diseases or disorders involving pathologic activation from C5a and non-pharmaceutical applications.
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priorityDate 2017-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56963851
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8FD60
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395633
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24821094
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381421502
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6992563
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP91850
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ69DK8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8FDU8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41687
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60667272
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID534492
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66612441
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41693
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451339314
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP18109
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381421641
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393647
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226789878
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281251
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381421645
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458392451
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID595146
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCJ9NSP1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56956742
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381421163
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCJ9P745
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID380373
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458392881
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395512
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4811496
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12600299
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP44309
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID192262
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415429153
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16410
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41683
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2897887
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1XHJ5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158927079
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395489
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16533
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507060
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5R960
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3LFK4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1494606
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403086
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396420
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9E8G2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4914
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395485
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68564
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID74048
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41522
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395428
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157250974
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04408
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395486
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1488261
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157250975
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1251836
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506776
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395488
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157250976
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9IRW3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397070
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCH9A0J9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2P902
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3KYH2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9WYN2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419517753
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID362119
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2PE47
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04363
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425890504
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1487533
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID58461422
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395413
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID629
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2PE78
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID43919
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41324
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395467
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP59437
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396778
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2VEX9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395468
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID644019
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396723
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5HMA3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6280
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506748
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581812
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID441335
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1486904
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11651
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29672699
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID498666
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506586
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8Y4A7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ66S64
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581866
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID57469701
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9WVG1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1487307
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68290
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID55590735
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1LGI7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID114447
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ66S65
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60901531
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCH0YYU7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68291
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41323
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID153274811
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1486634
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP42633
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID117027
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ865Y1

Total number of triples: 2023.