http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2020261450-A1

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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-54
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filingDate 2020-05-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7a11eca8e9680b9a546c8a0195efc677
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d34acc6c2e0473709d35f2b036b34d37
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1630d2a6842bd99ceb3a941bb10c42d4
publicationDate 2020-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2020261450-A1
titleOfInvention 6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE AS NEGATIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
abstract The present invention relates to novel 6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one derivatives as negative allosteric modulators (NAMs) of the metabotropic glutamate receptor subtype 2 (“mGluR2”). The invention is also directed to pharmaceutical compositions comprising such compounds, to processes for preparing such compounds and compositions, and to the use of such compounds and compositions for the prevention or treatment of disorders in which the mGluR2 subtype of metabotropic receptors is involved.
priorityDate 2014-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312184122
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312184114
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226476561
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10129899
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312181696
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ14BI2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID145787
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449794756
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157242840
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534566
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4L0Y3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227293359
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157854846
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449793880
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158580507
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157195183
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95106
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419567890
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118700113
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID240
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425623858
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70420125
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ02193
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432555903
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8148
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413668210
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1X707
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2904
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451711558
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1X706
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414839460
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29386
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1X705
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157892891
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID159898033
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1X704
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408848
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226489719
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24350
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1X703
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID567181
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447917096
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226478094
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1X702
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID446220
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226423208
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157247782
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID159253377
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158799131
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1X701
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136068742
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12460470
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1X700

Total number of triples: 681.