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publicationDate 2020-02-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2020038352-A1
titleOfInvention Co-crystals of nurr1-lbd in complex with a cyclopentenone prostaglandin and modulators of nurr1
abstract Co-crystals comprising the Nuclear receptor related 1 protein-ligand binding domain (Nurr1-LBD) and a cyclopentenone prostaglandin are provided. Also provided are methods of identifying or designing Nurr1-modulating ligands and compounds based on the crystal structures described herein as well as the applications of said ligands and compounds as Nurr1 modulators or medicaments.
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