http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2019314513-A1

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filingDate 2019-06-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_13066caa9d21419a8a5a776584b2a4a9
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_65ae4f1624b9657ad90c0775141d6fc7
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publicationDate 2019-10-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2019314513-A1
titleOfInvention Duocarmycin adcs showing improved in vivo antitumor activity
abstract The present invention relates to duocarmycin-containing antibody-drug conjugates (ADCs) for use in the treatment of human solid tumours and haematological malignancies expressing HER2, in particular breast cancer, gastric cancer, bladder cancer, ovarian cancer, lung cancer, prostate cancer, pancreatic cancer, colorectal cancer, head and neck squamous cell cancer or osteosarcoma, and acute lymphoblastic leukaemia. In particular, the present invention relates to duocarmycin-containing ADCs for use in the treatment of human solid tumours with HER2 IHC 2+ or 1+ and HER2 FISH negative tissue status. Advantageously, the present invention relates to duocarmycin-containing ADCs for use in the treatment of triple negative breast cancer (TNBC).
priorityDate 2014-01-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399456
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60953
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25591
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281740
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID443228
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9854073
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID146180348
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399572
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395836
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24337
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395835
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54278540
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6918289
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452922423
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733526
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID146179504
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226479495
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5994
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP70091
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID146179503
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4343013
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408415
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID20056954
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395879
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395878
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID454216
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136123990
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100009712
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4938396
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118655862
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6857599
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161023335
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399573
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID146179513
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1NRL7
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16740990
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396694
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID147887999
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395857
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66091
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP61110
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227125093
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID494003

Total number of triples: 348.