http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2019300503-A1

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filingDate 2017-06-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_83443b9d9c13716007a3b3ac900fc0d5
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publicationDate 2019-10-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2019300503-A1
titleOfInvention 5-[3-[piperazin-1-yl]-3-oxo-propyl]-imidazolidine-2,4-dione derivatives as adamts 4 and 5 inhibitors for treating e.g. osteoarthritis
abstract The present invention discloses compounds according to Formula I: n n n n n n n n n n Wherein R 1 , R 2 , R 3a , R 3b , R 6 , Cy, and the subscript n are as defined herein. n The present invention relates to compounds inhibiting ADAMTS, methods for their production, pharmaceutical compositions comprising the same, and methods of treatment using the same, for the prophylaxis and/or treatment of inflammatory diseases, and/or diseases involving degradation of cartilage and/or disruption of cartilage homeostasis by administering the compound of the invention.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2022212638-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2021158626-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2023011547-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-113754635-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-115052596-A
priorityDate 2016-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1749.