http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2019142963-A1

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filingDate 2017-04-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_89cbb3e7c75928c4b1cb7ca36b3140b2
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publicationDate 2019-05-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2019142963-A1
titleOfInvention Fgf21 c-terminal peptide optimization
abstract Disclosed herein are modified C-terminal fragments of FGF21 optimized for binding to Klotho β or antagonizing FGF21 activity. FGF21 peptides modified to comprise modifications to the C-terminal amino acid sequence are disclosed that have enhanced activity at the FGF21 receptor. Additionally, conjugates formed between the optimized FGF21 peptide fragments and insulin like peptides or nuclear hormone receptor ligands are provided.
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Total number of triples: 1843.