http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2019010154-A1

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filingDate 2016-07-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_45ba971efd38b7c74e7cb5f3494562f1
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_21fd7fbb79f28d9512cc7fed659169f6
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publicationDate 2019-01-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2019010154-A1
titleOfInvention Factor xia macrocycle inhibitors bearing a non-aromatic p2' group
abstract The present invention provides compounds of Formula (I): or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the variables are as defined herein. These compounds are selective factor XIa inhibitors or dual inhibitors of FXIa and plasma kallikrein. This invention also relates to pharmaceutical compositions comprising these compounds and methods of treating thromboembolic and/or inflammatory disorders using the same.
priorityDate 2015-07-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126545666
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420166647
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID77999
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID137379247
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10298
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381450981
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280833
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID137379242
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381451024
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126545664
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID137379240
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP33711
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381450996
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126545663
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID137379237
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID107378852
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381450995
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID282522
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A3Q1M7Q5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID137379236
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426124959
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381450994
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID137379223
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381450992
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408642107
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126545658
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID81782
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381450991
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426149262
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381450990
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413713178
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100356068
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126545674
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID381450989
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID168937
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396834
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394749
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126545672
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A2R6Q324
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419521555
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394949
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396796
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP34006
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12910406
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5702640
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3806790
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP34005
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311722830
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID229605644
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419563342
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6166165

Total number of triples: 1628.