http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2018356395-A1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_7bee2f1c3fb5dd643bf0d19863df0b0a
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/G01N2500-10
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/G01N33-502
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/G01N33-5026
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/G01N33-50
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filingDate 2018-06-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fd9d6daec91423a5e4fa33b649fcf654
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_53aca7a9db12e15b5515abf55fdde507
publicationDate 2018-12-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2018356395-A1
titleOfInvention Compounds and methods of identifying, synthesizing, optimizing and profiling protein modulators
abstract This invention relates to methods of identifying, synthesizing, optimizing and profiling compounds that are inhibitors or activators of proteins, both naturally occurring endogenous proteins as well as certain variant forms of endogenous proteins, and novel methods of identifying such variants. The method accelerates the identification and development of compounds as potential therapeutically effective drugs by simplifying the pharmaceutical discovery and creation process through improvements in hit identification, lead optimization, biological profiling, and rapid elimination of toxic compounds. Implementation results in overall cost reductions in the drug discovery process resulting from the corresponding increases in efficiency.
priorityDate 2005-05-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1398.