http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2018339982-A1

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filingDate 2018-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_52519511ac8ec7224c447bbba15f13ef
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_85c73def63c055f072a36a12609adbe1
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publicationDate 2018-11-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2018339982-A1
titleOfInvention Bicyclic heterocyclic derivatives as bromodomain inhibitors
abstract The present disclosure provides bicyclic heterocyclic derivatives of formula (I), which may be therapeutically useful, more particularly as bromodomain inhibitors; (I), in which R 1 , R 2 , R 3 , R 4 , L 1 , L 2 , Cy 1 , Cy 2 , X, n, and dotted line have the same meaning given in the specification, and pharmaceutically acceptable salts or pharmaceutically acceptable stereoisomers thereof that are useful in the treatment and prevention of diseases or disorders, in particular their use in diseases or disorders associated as bromodomain inhibitors. The present disclosure also provides preparation of compounds and pharmaceutical formulations comprising at least one of bicyclic heterocyclic derivatives of formula (I), together with a pharmaceutically acceptable carrier, diluent, or excipient.
priorityDate 2014-01-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66774101
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450767085
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID230539927
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157601577
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118224582
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656724
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311660604
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118224579
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656726
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311660541
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656722
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311660567
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID229928816
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656723
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394040
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450670696
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID237841968
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656729
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158306142
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14489769
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226428638
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID79792
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656730
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226517933
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157582464
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID124137246
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656727
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23676152
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226447673
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394094
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656728
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311660453
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9838
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409038092
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID10566
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453917849
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656715
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311660477
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453631720
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656717
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453923783
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226593741
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311660422
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161812409
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311660502
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID229183392
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID85702122
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311660509
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135385273
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID521435
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450560848
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID311660487
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID124137024
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID85702142
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89345217
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394012
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11776
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433409228
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7018254
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656711
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450505166
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID522490
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID329656712

Total number of triples: 994.