http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2018148469-A1

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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a582311bf84146893c583b5a1790151b
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publicationDate 2018-05-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2018148469-A1
titleOfInvention Process for preparation of sulfonylurea bile acid derivatives
abstract The present invention relates to processes for preparing a compound of Formula I: n n n n n n n n n n or a pharmaceutically acceptable salt or solvate thereof. These compounds and pharmaceutical compositions are useful as FXR or TGR5 modulators. Specifically, the present invention relates to bile acid derivatives and methods for their preparation and use. n The present invention relates to a process for the preparation of a compound (II) and its salts and derivatives which are useful intermediates in the synthesis of biologically active molecules, especially in the synthesis of FXR and TGR5 modulators. n n n n n n n n n n The present invention also relates to a process for the preparation of a compound (III) and its diethylamine salt.
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373686
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393257
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393245
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71832
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6274
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID994
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2723939
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415027654
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395715
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226394498
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69466
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID436847
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21491
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2724141
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60351
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID791
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO18531
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID374822803
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID374818254
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448285482
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1148
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID374822790
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID160213804
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID76328184
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5359272
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2641
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8818
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393392
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID985
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Total number of triples: 415.