http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2018134709-A1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_da69597f7db360db56f35351150d305c
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02A50-30
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D473-34
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D473-34
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00
filingDate 2016-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1f6b5c2563d2f4719de5228eddf6b00b
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6dd17b79085131a5a8e58b3b64da7da2
publicationDate 2018-05-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2018134709-A1
titleOfInvention Purinyl-n-hydroxyl pyrimidine formamide derivative, preparation methods and uses thereof
abstract The present invention relates to the field of the chemical medicines, and in particular, to purinyl-N-hydroxyl pyrimidine formamide derivatives, a preparation method therefor and a use thereof. The present invention provides a purinyl-N-hydroxyl pyrimidine formamide derivative having a structure represented by formula (I). The invention also provides a method for preparing said purinyl-N-hydroxyl pyrimidine formamide derivative and a use thereof. Purinyl-N-hydroxyl pyrimidine formamide derivative provided in the invention can be not only a PI3K and HDAC double-functional target kinase inhibitor, but also a PI3K or HDAC single target kinase inhibitor, thus providing new choice for preparing multi-target inhibitors.
priorityDate 2015-04-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 927.