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filingDate 2015-10-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6d63dabc07faa24d5e1ade30510419a1
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publicationDate 2018-01-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2018022730-A1
titleOfInvention Small-molecule inhibitors targeting discoidin domain receptor 1 and uses thereof
abstract Compounds of formula (I), their pharmaceutically acceptable salts and stereoisomers thereof, as well as application in effectively inhibiting the enzymatic activity of discoidin domain receptor 1 and can be used as new therapeutic agents for preventing and treating e.g. inflammation, liver fibrosis, kidney fibrosis, lung fibrosis, skin scar, atherosclerosis, and cancer. The compound of formula I is: wherein the variables are as defined herein.
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priorityDate 2014-10-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 1699.