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publicationDate 2017-01-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2017001950-A1
titleOfInvention COMPOUNDS FOR TARGETING DRUG DELIVERY AND ENHANCING siRNA ACTIVITY
abstract Here described are compounds consisting of the structuren (targeting molecule) m -linker-(targeting molecule) n ,n nwherein the targeting molecule is a retinoid or a fat soluble vitamin having a specific receptor on the target cell; wherein m and n are independently 0, 1, 2 or 3; and wherein the linker comprises a polyethylene glycol (PEG) or PEG-like molecule, as well as compositions and pharmaceutical formulations including these compounds which are useful for the targeting and delivery of therapeutic agents; and methods of using these compositions and pharmaceutical formulations.
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Total number of triples: 771.