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publicationDate 2016-10-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2016303084-A1
titleOfInvention Diazole lactams
abstract Compounds are provided that act as potent antagonists of the CCR1 receptor, and have in vivo anti-inflammatory activity. The compounds are diazole lactam derivatives and are useful in pharmaceutical compositions, methods for the treatment of CCR1-mediated disease, and as controls in assays for the identification of competitive CCR1 antagonists.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90215451
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5J732
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Total number of triples: 1369.