http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2016008486-A1

Outgoing Links

Predicate Object
assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_4fede5e271fe9a3788b900c0ce6e0054
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K2317-24
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K2317-76
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K2039-505
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K39-3955
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K16-40
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6801
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6803
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K16-32
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-60
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K16-30
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6889
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6855
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6851
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6863
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6871
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6809
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-6849
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K47-48646
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-19
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-437
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-05
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-02
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K45-06
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-48
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K16-40
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K45-06
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K39-395
filingDate 2015-09-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_13066caa9d21419a8a5a776584b2a4a9
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a717adcffb5e13ae8257ab9d574568c1
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4dc59e3a9daf8413a408c014acdc5433
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_65ae4f1624b9657ad90c0775141d6fc7
publicationDate 2016-01-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2016008486-A1
titleOfInvention Duocarmycin adcs showing improved in vivo antitumor activity
abstract The present invention relates to duocarmycin-containing antibody-drug conjugates (ADCs) for use in the treatment of human solid tumours and haematological malignancies expressing HER2, in particular breast cancer, gastric cancer, bladder cancer, ovarian cancer, lung cancer, prostate cancer, pancreatic cancer, colorectal cancer, head and neck squamous cell cancer or osteosarcoma, and acute lymphoblastic leukaemia. In particular, the present invention relates to duocarmycin-containing ADCs for use in the treatment of human solid tumours with HER2 IHC 2+ or 1+ and HER2 FISH negative tissue status. Advantageously, the present invention relates to duocarmycin-containing ADCs for use in the treatment of triple negative breast cancer (TNBC).
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9629924-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-11052155-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9901567-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9815784-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10266606-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2020205986-A1
priorityDate 2014-01-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

Incoming Links

Predicate Subject
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2009010945-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2012214864-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2013095172-A1
isDiscussedBy http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126941
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395485
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID115369
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60750
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458033181
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396322
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284616
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399747
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31703
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396105
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450540726
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57300161
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID36314
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226403436
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID114361
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395471
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID576940
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399177
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226403435
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226470237
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226521722
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119691
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161023335
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395836
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396787
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID136123990
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399412
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2187
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312138810
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60700
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118655863
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135565230
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395835
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312138816
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226443492
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396057
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5394
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312138807
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227959075
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2907
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6274
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399366
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453916508
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71384
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226525567
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158815302
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400582
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414353776
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227125093
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12233
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396694
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148124
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399253
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226393819
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5865
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID454216
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399254
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448084636
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312138809
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449808904
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60198
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226523119
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID30323
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID159344117
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395766
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87072684
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID20056954
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57504783
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13183883
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID228389233
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57129391
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7427
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161707418
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452922423
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420256212
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408415
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13316162
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID149404705
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID208908
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399616
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21158526
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395940
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID773
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15943264
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID64780
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226400014
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447680698
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID231737968
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226397750
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6442177
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID123631
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227081507
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399573
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312138815
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733526
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4112
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399572
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396419
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458033180
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6251
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19875453
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118655862
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399016
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396417
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4634576
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID104741
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3902
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3032583
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395318
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4212
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60838
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4126408
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21714437
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID227080867
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396389
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157531530
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3690
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395632
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399858
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157219484
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135410875
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396147
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399457
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226468634
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226522492
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148325014
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5311497
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13342
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5994
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14746059
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410770558
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396146
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399456
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395878
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID235516
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395879
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135403648
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5312965
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226407884
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396349
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226404269
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395512
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396360
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID312138808
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118655856
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID176870
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60953
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395857
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118655857
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161418836
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453496208
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID41867
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395292
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395486

Total number of triples: 204.