http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2015315183-A1

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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K45-06
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filingDate 2013-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a37b51be7ba770b4c02acc54b226a04b
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4042123fb012d38d20e144a193c5470b
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d9f2a42c29b754973679937d08c7fff6
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_68f11a90c8161936ba66dcae7ffb279b
publicationDate 2015-11-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2015315183-A1
titleOfInvention Novel octahydropyridoquinazoline derivative, pharmaceutical composition containing same, and uses for said deriavative and composition
abstract [Problem] To provide a novel compound that exhibits an agonistic effect on dopamine D 2 receptors. n [Solution] The present invention provides a compound represented by the general formula (I): n n n n n n n n n n in which R 1 is C 1-6 alkyl or the like; R 2 is hydrogen or the like; R 3 and R 4 are each hydrogen, C 1-6 alkyl, R 10 R 11 N—C 1-6 alkyl, aralkyl, or the like; R 5 and R 6 are hydrogen or the like; and R 7 is hydrogen or the like, or a pharmaceutically acceptable salt thereof, a pharmaceutical compositions containing same and uses for said compound/salt and composition. The compounds of the present invention exhibit potent dopamine D 2 receptor simulating activities and thus are useful as a treating or preventing agent for Parkinson's disease and the like.
priorityDate 2012-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1351.