http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2015141457-A1

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_1a615b6db0acb71ee30f71f157888ba2
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-146
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-47
filingDate 2013-05-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f02e6d61a214939698206afd721cdaa6
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c12c6815af885117b3514cdb7765cae2
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a0e066f2accd3ce7b492101fd3dc5000
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c44569476f0fa8935859f1032fc4cee0
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d16ab1ef4dec38cc90397afffacc09e6
publicationDate 2015-05-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2015141457-A1
titleOfInvention Elvitegravir solid dispersion
abstract The present invention provides a novel amorphous solid dispersion of elvitegravir in combination with a pharmaceutically acceptable carrier, process for its preparation and pharmaceutical compositions comprising it. In a preferred embodiment the process for the preparation of amorphous solid dispersion of elvitegravir in combination with a pharmaceutically acceptable carrier comprises: preparing a solution comprising a mixture of elvitegravir and one or more pharmaceutically acceptable carriers selected from copovidone, ethyl cellulose, hydroxypropyl methylcellulose, polyethylene glycol, span 20 or soluplus in a solvent; and removing the solvent from the solution obtained; adding hydrocarbon solvent to the residual solid; and isolating amorphous solid dispersion of elvitegravir in combination with a pharmaceutically acceptable carrier.
priorityDate 2012-05-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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