http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2014288133-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-06
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-14
filingDate 2014-06-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4e8383ab09633ade08181465cd353254
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a9a64820367b3c2fd9fe108e75a31fd2
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_75113504340d563e4d935a20b9e863f0
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1a3f71bbac590084ae3a713c62211409
publicationDate 2014-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2014288133-A1
titleOfInvention 3 -amino- pyrazole derivatives useful against tuberculosis
abstract A compound of Formula (I) or a pharmaceutically acceptable salt thereof: n n n n n n n n n n Wherein: Het is a 5 to 10-membered heteroaromatic ring; Either X is N and Y is CR 5 ; or X is C and Y is S; Z is selected from N and CH; R 1 is selected from H and C 1-2 alkyl; R 2 is selected from H, C 1-2 alkyl, OH, —CH 2 OH and C 1-2 alkoxy; Each R 3 is independently selected from OH, C 1-3 alkyl, F, Cl, Br, NH 2 , and C 1-3 alkoxy; R 4 is selected from C 1-3 alkyl and haloC 1-3 alkyl; R 5 is selected from H, C 1-3 alkyl and haloC 1-3 alkyl; R 6 and R 7 are either i) each independently selected from H, C 1-3 alkyl and C 1-3 alkoxy; or ii) R 6 and R 7 together with the ring to which they are attached form a 9-membered bicylic ring; p is 0-3; and R A is selected from H and C 1-3 alkyl, compositions containing them, their use in therapy, for example in the treatment of tuberculosis, and methods for the preparation of such compounds, are provided.
priorityDate 2010-10-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 2100.