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filingDate 2012-10-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0018c6303f1b1ec842e02aee6a349f04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_41b0e97ab9fc9f35a408de75f8e98353
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publicationDate 2014-09-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2014275097-A1
titleOfInvention NOVEL CHIRAL N-ACYL-5,6,7(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
abstract The present invention relates to novel compounds of Formula I and their use in therapeutic treatments. The invention further relates to a novel chiral synthesis of 5,6,7,(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines using N-sp3 protective groups. The invention also provides intermediates for use in the synthesis of compounds of Formula I.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9987274-B2
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID78108063
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID567306
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID239819722
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458108599
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID323504923

Total number of triples: 1238.