http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2014235537-A1

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filingDate 2012-08-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1742104c25b6763728d674470d2e4c00
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publicationDate 2014-08-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2014235537-A1
titleOfInvention N-glycosylated insulin analogues
abstract Compositions and formulations comprising N-glycosylated insulin analogues are described. In particular embodiments, the glycosylated insulin analogues are produced in vivo and comprise one or more the N-linked N-glycans selected from high mannose or fucosylated or non-fucosylated hybrid, paucimannose, or complex N-glycans. In other embodiments, the N-glycan comprising the high mannose or fucosylated or non-fucosylated hybrid, paucimannose, or complex N-glycan is attached to the insulin analogue in vitro. Examples of N-glycans include but are not limited to a molecule having a structure selected from N-glycans in the group consisting of Man( 1 — 9 )GlcNAc 2 ; or selected from N-glycans in the group consisting of GlcNAc (1 — 4) Man 3 GlcNAc 2 ; or selected from N-glycans in the group consisting of Gal(j. 4)GlcNAc (1 — 4) Man 3 GlcNAe 2 ; or selected from N-glycans in the group consisting of NANA({umlaut over (ι)}_4)Gal (1 — 4) GlcN Ac (1 — 4) Man 3 GlcN Ac 2 —
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Total number of triples: 1409.