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publicationDate 2014-03-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2014072558-A1
titleOfInvention Activin Receptor Type II B Inhibitors Comprising DLK1 Extracellular Water-Soluble Domain
abstract The present invention relates to an activin receptor type II B (ACVR2B) inhibitor which comprises the delta-like 1 homolog (DLK1) extracellular water-soluble domain. More specifically, the present invention relates to an extracellular soluble domain of DLK1; fragments of the extracellular soluble domain of DLK1; mutants of the extracellular soluble domain of DLK1; a composition for suppressing ligand linkage with the ACVR2B receptor, which includes a fragment of the mutants as an active ingredient; and a pharmaceutical composition for prevention and treatment of diseases which comprises the same. The composition of the present invention competitively binds to the ACVR2B receptor and inhibits the binding of an ACVR2B ligand to the ACVR2B receptor, which inhibits protein signalling associated with such ligands, and will be useful for prevention and treatment of diseases associated therewith.
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9WS40
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID81822
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1NNP2
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9W7R2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ77IS8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ77E03
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO35312
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID421931
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP16285
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19691
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24378
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID517541
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8BCV5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11212
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8B6J9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11211
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID728378
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19534
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID476196
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ66453
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID39130
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25644
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24304
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07453
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6J1J2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID420868
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6868
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8AVB2
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID43826
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8B0H9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ07097
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID64083
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ20EU8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81025
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO76745
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID631990
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO14793
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6032
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCCAA54692
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ06SH2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP03521
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95J86
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1KVQ9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407024245
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53784538
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29152
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19022
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID617566
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ86523
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ03332
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12162
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID83729
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3875052
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID30291
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5K2K7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11491
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2064
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ90275
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68245
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68243
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8UWD9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27371
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID30639
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID326282
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8UWD8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12161
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DOF3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID10220
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8V3T7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP29335
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ86134
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ65111
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID85272
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6XGL2
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP18075
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16326
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID459018
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID535916
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395247
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100037061
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5959
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23359
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID91
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6X5V1
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO55075
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A286ZV08
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41522
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Total number of triples: 469.