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filingDate 2011-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2013-08-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2013209390-A1
titleOfInvention Process For Producing Drug-Block Copolymer Composite And Pharmaceutical Preparation Containing Same
abstract [Problem] There has been a requirement for a process for producing a pharmaceutical preparation that is obtained by encapsulating a uniform poorly water-soluble drug in a block copolymer, and dissolves immediately with an addition of water, and does not contain residues of organic solvents. n [Solution] Provided is a method for producing a drug-block copolymer composite, the method comprising: mixing a poorly water-soluble drug and a block copolymer including a hydrophilic segment and a hydrophobic segment bonded together, in one or more non-aqueous solvents; optionally heating the mixture as necessary; and spray-drying the resulting mixture liquid.
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