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filingDate 2010-10-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_dc5d01d10069d1e61d454d5add31a273
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6f70f807717d5e63d2895cec7f626848
publicationDate 2013-08-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2013203988-A1
titleOfInvention Process for making bortezomib and intermediates for the process
abstract The invention relates to processes of making bortezomib of formula (1) enantiomers thereof and/or intermediates thereof, comprising at least one step of coupling a carboxylic acid with an amine, wherein the coupling step is performed in a presence of the compound of formula (8), wherein A is C1-C6 alkyl group, preferably wherein A is n-propyl group.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-103374026-A
priorityDate 2010-10-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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