http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2013079339-A1

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filingDate 2010-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_86e642199c6bc172d41338fae2225bea
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publicationDate 2013-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2013079339-A1
titleOfInvention Trpv1 vanilloid receptor antagonists with a bicyclic portion
abstract The invention discloses compounds of formula I n n n n n n n n n n n n wherein Y is a group of formula A, B, C, D, or E: n n n n n n n n n n n n n n n n and W, Q, n, R1, R2, R3, U1-U5, J and K have the meanings given in the description. n n n n n The compounds of formula I are TRPV1 antagonists and are useful as active ingredients of pharmaceutical compositions for the treatment of pain and other conditions ameliorated by the inhibition of the vanilloid receptor TRPV1.
priorityDate 2010-03-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1091.