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filingDate 2012-04-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8485d293e1fb801f424a3a814f96d4eb
publicationDate 2012-11-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2012289471-A1
titleOfInvention Novel compounds with high therapeutic index
abstract The present invention is directed to novel therapeutic compounds comprised of an amino acid bonded to a medicament or drug having a hydroxy, amino, carboxy or acylating derivative thereon. These high therapeutic index derivatives have the same utility as the drug from which they are made, and they have enhanced pharmacological and pharmaceutical properties. In fact, the novel drug derivatives of the present invention enhance at least one therapeutic quality, as defined herein. The present invention is also directed to pharmaceutical compositions containing same.
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Total number of triples: 3023.