http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2012225907-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-454
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filingDate 2012-05-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_cdd141ec7fa963be0553298708b1b488
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fe629ab2ed9e88b59ab53c170f6a4193
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publicationDate 2012-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2012225907-A1
titleOfInvention Benzamide compounds useful as histone deacetylase inhibitors
abstract The invention concerns benzamide compounds of formula (I): compound of formula (I): n n n n n n n n n n wherein R 1 is a C-linked pyrazole ring, which is optionally substituted by one or more groups selected from C 1-4 alkyl, C 3-4 cycloalkyl, C 1-4 alkoxy and C 3-4 cycloalkoxy;n nor a pharmaceutically acceptable salt or pro-drug form thereof. The invention also concerns processes for the preparation of such compounds, pharmaceutical compositions containing them and their use in the manufacture of a medicament for use as an antiproliferative agent in the prevention or treatment of tumours or other proliferative conditions, which are sensitive to the inhibition of histone deacetylase (HDAC).
priorityDate 2005-10-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1251.