http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2012129890-A1

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filingDate 2010-07-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b46d0108999bfb28882fa6ab62ef3cd3
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6466fbfb5bea9b5b32d73cc07e0f936a
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publicationDate 2012-05-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2012129890-A1
titleOfInvention Indole derivative or pharmaceutically acceptable salt thereof
abstract A compound (I) of the present invention, which has an EP 1 receptor antagonism: n n n n n n n n n n n n [wherein A represents a benzene ring or the like; Y 1 represents a C 1-6 alkylene group; Y 2 represents a single bond or the like; R 1 represents a hydrogen atom, a C 1-6 alkyl group or the like; R 2 represents a phenyl group which may have a substituent, a 5-membered aromatic heterocyclic ring which may have a substituent, a 6-membered aromatic heterocyclic ring which may have a substituent or the like; R 3 represents a halogen atom, a C 1-6 alkoxy group or the like; R 4 represents a hydrogen atom or the like; and R 5 represents a hydrogen atom or the like] or a pharmaceutically acceptable salt thereof is provided. Furthermore, the compound (I) of the present invention can be used as an agent for treating or preventing LUTS, in particular, various symptoms of OABs.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-8815903-B2
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priorityDate 2009-07-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 3071.