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filingDate 2010-04-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8852e0de29ac2a22ed77659fbf4b833c
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publicationDate 2012-04-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2012094996-A1
titleOfInvention Imidazo [2, 1-B] [1, 3, 4] Thiadiazole Derivatives
abstract There is provided compounds of formula (I): wherein R 1 , R 2 and R 3 have meanings given in the description, and pharmaceutically-acceptable esters, amides, solvates or salts thereof, which compounds are useful in the treatment of diseases in which inhibition of a protein or lipid kinase (e.g. PI3-K, particularly class I PI3K) is desired and/or required, and particularly in the treatment of cancer.
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Total number of triples: 1328.