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filingDate 2011-02-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1b0754aba48fc861c739c7e1acbf1a4b
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publicationDate 2012-02-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2012041190-A1
titleOfInvention Macrocycles as factor xia inhibitors
abstract The present invention provides compounds of Formula (I): n n n n n n n n n n or a stereoisomer, a tautomer, or a pharmaceutically acceptable salt thereof, wherein all the variables are as defined herein. These compounds are selective Factor XIa inhibitors or dual inhibitors of fXIa and plasma kallikrein. This invention also relates to pharmaceutical compositions comprising these compounds and methods of treating thromboembolic and/or inflammatory disorders using the same.
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priorityDate 2010-02-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408138716
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226795327
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID455678035
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408161108
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID107428
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID88581181
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396246
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128537407
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID324110592
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407933440
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128768619
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396247
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128809644
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408007536
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8406
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396248
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID88581241
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408017724

Total number of triples: 7193.