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filingDate 2011-10-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3efd23428ecf201af1ee7a18af301f00
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publicationDate 2012-02-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2012040982-A1
titleOfInvention Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions
abstract The present invention relates to substituted xanthines of general formula n n n n n n n n n n wherein R 1 to R 4 are as defined herein, the tautomers and the stereoisomers thereof, mixtures thereof, the prodrugs and the salts thereof which have valuable pharmacological properties, particularly an inhibiting effect on the activity of the enzyme dipeptidylpeptidase-IV (DPP-IV).
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Total number of triples: 5857.