http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2011306563-A1

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filingDate 2009-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_01ab05805460b0b1812a40663a5dc18c
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publicationDate 2011-12-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2011306563-A1
titleOfInvention Macrolactone derivatives, method for the production thereof and use thereof for the treatment of cancer
abstract The present invention relates to the use of a compound of the formula (I), wherein X and Y independently of one another are OH, O—(C 1 -C 6 )-alkyl, NH 2 or NH—(C 1 -C 6 )-alkyl, or X and Y together form a group —O— or wherein X and Y together form a further bond between the C atoms to which they are attached; R1 and R2 independently of one another are H, Cl or Br; R3 is H,(C 1 -C 6 )alkyl, C(═O)—(C 1 -C 6 )-alkyl or (C 1 -C 6 )-alkylene-NH—(C 1 -C 6 )-alkyl; R4 is H, (C 1 -C 6 )-alkyl or C(═O)—(C 1 -C 6 )-alkyl, and R5 is methyl or ethyl; or a physiologically tolerable salt of a compound of the formula (I), for the treatment and/or prophylaxis of cancer diseases, a pharmaceutical composition for the treatment and/or prophylaxis of cancer diseases comprising a compound of the formula (I), a compound of the formula (I) and a process for the preparation of the compound (I).
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-114605430-A
priorityDate 2008-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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