http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2011236367-A1

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filingDate 2010-05-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f75d298f5562d8e29fb9a71de4954a0d
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publicationDate 2011-09-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2011236367-A1
titleOfInvention Rat cathespin dipeptidyl peptidase i (dppi): crystal structure and its uses
abstract The present invention relates to structural studies of dipeptidyl peptidase I (DPPI) proteins, modified dipeptidyl peptidase I (DPPI) proteins and DPPI co-complexes. Included in the present invention is a crystal of a dipeptidyl peptidase I (DPPI) and corresponding structural information obtained by X-ray crystallography from rat and human DPPI. In addition, this invention relates to methods for using structure co-ordinates of DDPI, mutants hereof and co-complexes, to design compounds that bind to the active site or accessory binding sites of DPPI and to design improved inhibitors of DPPI or homologues of the enzyme.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-109988228-A
priorityDate 2000-09-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 424.