http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2011166162-A1

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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_61beac9e03d80617d92ad25cb991d447
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publicationDate 2011-07-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2011166162-A1
titleOfInvention 1,2-Benzisothiazole Compounds Useful for Combating Animal Pests
abstract The present invention relates to sulfonamide compounds of formula (I) n n n n n n n n n n wherein R 1 is H, halogen, CN, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 7 -cycloalkyl, C 3 -C 7 -cycloalkyl-C 1 -C 4 -alkyl, C 1 -C 6 -alkoxy, C 2 -C 6 -alkenyloxy, C 2 -C 6 -alkynyloxy, C 1 -C 6 -alkylthio, C 2 -C 6 -alkenylthio, C 2 -C 6 -alkynylthio, C 1 -C 6 -haloalkyl or C 1 -C 6 -haloalkoxy; R 2 and R 3 are H, halogen, CN, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 7 -cycloalkyl, C 3 -C 7 -cycloalkyl-C 1 -C 4 -alkyl, C 1 -C 6 -alkoxy, C 2 -C 6 -alkenyloxy, C 2 -C 6 -alkynyloxy, C 1 -C 6 -alkylthio, C 2 -C 6 -alkenylthio, C 2 -C 6 -alkynylthio, C 1 -C 6 -haloalkyl or C 1 -C 6 -haloalkoxy; or R 2 together with R 3 form a fused 5 or 6-membered carbocycle or heterocycle; R 4 is halogen, CN, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 1 -C 6 -alkoxy, C 1 -C 6 -alkylthio, C 1 -C 6 -alkylsulfinyl, C 1 -C 6 -alkylsulfonyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -haloalkoxy, C 1 -C 6 -haloalkylthio, C 1 -C 6 -haloalkylsulfinyl or C 1 -C 6 -haloalksulfonyl; n is 0, 1, 2 or 3; R 5 is phenyl or a 5- or 6-membered heterocycle; X is O or NR x , wherein R x is H, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 7 -cycloalkyl, C 1 -C 6 -alkoxy, C 2 -C 6 -alkenyloxy, C 2 -C 6 -alkynyloxy, C 1 -C 6 -alkylcarbonyl or C 1 -C 6 -alkylcarbonyloxy; Y is N or C(R y ), wherein R y is H, halogen, CN, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 7 -cycloalkyl, C 3-7 -cycloalkyl-C 1 -C 4 -alkyl, C 1 -C 6 -alkoxy, C 2 -C 6 -alkenyloxy, C 2 -C 6 -alkynyloxy, C 1 -C 6 -alkylthio, C 2 -C 6 -alkenylthio, C 2 -C 6 -alkynylthio, C 1 -C 6 -haloalkyl and C 1 -C 6 -haloalkoxy; and Z is a chemical bond, O or N(R z ), wherein R z is C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 7 -cycloalkyl, C 1 -C 6 -alkoxy, C 2 -C 6 -alkenyloxy, C 1 -C 6 -alkylcarbonyl or C 1 -C 6 -alkylcarbonyloxy;n nas well as to the N-oxides and salts thereof. These compounds are useful for combating animal pests. The invention also relates to a process for the preparation of these compounds and to intermediate compounds used in said process. The invention further relates to a method for controlling animal pests by using the compounds of formula (I), the N-oxides or the salts thereof, to plant propagation material and to an agricultural and veterinary composition comprising said compounds, the N-oxides or the salts thereof.
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Total number of triples: 4407.