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filingDate 2010-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a44b890df55b26e71b1ee1275387cbee
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5611a9942a60e88de848e428233fa268
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_55e9fe1f4012e591369d6e1a53c24e03
publicationDate 2011-02-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2011034481-A1
titleOfInvention Novel tetrahydroisoquinoline derivative
abstract The present invention relates to a compound or a pharmacologically acceptable salt thereof having an excellent DGAT inhibitory effect and feeding suppressant effect. The present invention provides a compound represented by the general formula (I), or pharmacologically acceptable salt thereof: n n n n n n n n n n [wherein,n R 1 represents a phenylaminocarbonyl group that may be substituted with 1 to 5 group(s) independently selected from Substituent Group A, a benzoxazol-2-yl group that may be substituted with 1 to 3 group(s) independently selected from Substituent Group A, or the like; R 2 independently represents a C 1 -C 6 alkyl group; R 3 represents a group represented by the formula —C(═O)—O—R 4 or the like; R 4 represents a hydrogen atom, a C 1 -C 6 alkyl group that may be substituted with 1 to 3 group(s) independently selected from Substituent Group B, or the like; X represents an oxygen atom, a methylene group, or a group represented by the formula —NH—, or the like; L represents a single bond, a methylene group, or the like; . . . represents a single bond or a double bond; m represents 1 or 2; n represents an integer of 0 to 5; Substituent Group A represents a halogen atom, a C 1 -C 6 alkyl group, a C 1 -C 6 halogenated alkyl group, a C 1 -C 6 alkoxy group, or the like; and Substituent Group B represents a C 3 -C 6 cycloalkyl group, a phenyl group, a carboxyl group, or the like].
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2011152282-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2012202847-A1
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http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9216964-B2
priorityDate 2008-03-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 3520.