http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2010234601-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-04
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filingDate 2009-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7e322f1bc485605a2e508262ceeeeef3
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3baa0e8cb58bf592f212ba72d7e5f64a
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publicationDate 2010-09-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2010234601-A1
titleOfInvention Transition metal catalyzed synthesis of 2H-indazoles
abstract The present invention relates to a process for the regioselective synthesis of compounds of the formula I, n n n n n n n n n n wherein R0; R1; R2; R3; R4; R5; A1; A2; A3; A4, Q and J have the meanings indicated in the claims. The present invention provides a direct transition metal catalyzed process to a wide variety of multifunctional 2H-indazoles or 2H-azaindazoles of the formula (I) from 2-halo-phenylacetylenes or (2-sulfonato)phenylacetylenes and monosubstituted hydrazines.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10538603-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-10723818-B2
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9487506-B2
priorityDate 2007-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1187.