http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2010063084-A1

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00
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filingDate 2009-11-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_523ae4aebf61eb93f59e8fed451f7519
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3ee0e4cc6161b0ef05fb641a6e5f415d
publicationDate 2010-03-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2010063084-A1
titleOfInvention Multi-phase release methscopolamine compositions
abstract Formulations have been developed administering methscopolamine in multi-phases. In a preferred embodiment, the formulation contains methscopolamine in an immediate release. (“IR”) form and a sustained or delayed release (“DR”) form and/or poised release (“PR”) form. In another embodiment, the methscopolamine is released in a gradient, decreasing the side effects associated with rapidly elevated blood levels. In another embodiment the drug is bound to an ion-exchange resin, which can be suspended in a liquid or incorporated into a matrix for delayed, sustained and/or pulsed release. Dosage unit forms may be tablets, gels, liquids, capsules, beads, microparticles, films or lozenges. Multi-phase delivery can also be achieved through the use of a kit that provides for dosage escalation. This kit can be a blister pack or equivalent, wherein the drug is packaged so that a first dosage is taken, then sequentially larger dosages. The dosages can be the same in each unit, and instructions provided so that the correct dosage is obtained through the number of units and the time of administration or the dosages may be different, and the units ordered so dial the desired dosage administration profile is obtained when the patient takes the units in order as instructed.
priorityDate 2006-09-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129335952
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396388
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226420658
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129225114
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128018039
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID155366
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127944725
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4762
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226420683
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396789
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226413768
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3291
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226409030
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399399
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129503949
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5HKP6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226420720
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128692968
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4760
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284543
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396326
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226424261
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5566
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID136080371
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53627474
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5556
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4075
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226454824
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129082949
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129160840
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31205
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399472
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226406050
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21863265
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226425808
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129083571
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226412294
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID249343666
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4095
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226412295
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284566
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127729747
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127378182
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226406099
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID136088414
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226406100
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226406583
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284570
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396472
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5974
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4781
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66583097
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23897
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID181817
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226406509
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5984
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID92943

Total number of triples: 991.