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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7ede1565c01960d27ebf9dc4f6f036ea
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publicationDate 2009-10-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2009270433-A1
titleOfInvention 2,3-dihydro-iminoisoindole derivatives
abstract A compound represented by the following general formula (1), or a salt thereof has serine protease inhibiting activity, and particularly excellent inhibiting activity against clotting factor VIIa. This compound or a salt thereof is useful as therapeutic and/or prophylactic agents for diseases associated with thrombus formation. n n n n n n n n n n [wherein R 1 represents hydrogen, R 2 represents optionally substituted phenyl, etc., R 3 represents optionally substituted C6-10 aryl, etc.]
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Total number of triples: 2074.