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filingDate 2007-07-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2009-10-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2009253673-A1
titleOfInvention Substituted Pyrazoles as Ghrelin Receptor Antagonists
abstract Certain novel N-acylated spiropiperidine derivatives are ligands of the human ghrelin receptor(s) and, in particular, are antagonists/inverse agonists of the human ghrelin receptor. They are therefore useful for the treatment, control, or prevention of diseases and disorders responsive to the modulation of the ghrelin receptor, such as obesity, diabetes, and metabolic syndrome.
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Total number of triples: 4338.