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publicationDate 2009-07-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2009175888-A1
titleOfInvention Methods of treating cancer with an antibody-drug conjugate
abstract The present invention provides analogues of duocarmycins that are potent cytotoxins. Also provided are peptidyl and disulfide linkers that are cleaved in vivo. The linkers are of use in forming prodrugs and conjugates of the cytotoxins of the invention as well as other diagnostic and therapeutic moieties. The invention provides prodrugs and conjugates of the duocarmycin analogues with the linker arms of the invention.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226399399
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226658528
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID243505936
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID335929
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID138985298
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127931844
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID138985276
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID248442337
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135398679
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID138985273
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID142289861
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID138985274
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226408555
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57098364
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID138985279
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226664672
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127733291

Total number of triples: 935.