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filingDate 2007-07-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_65366ca74ad526a9c33ed834fdd37ec5
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publicationDate 2009-05-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2009118309-A1
titleOfInvention Selective antagonists of A2A adenosine receptors
abstract The present invention provides compounds of formulae Ia and Ib: n n n n n n n n n n wherein R 1-5 , Q, X, Y, Z, p, q, and r are as defined herein. The compounds are potent and selective antagonists of A 2A adenosine receptors (ARs). The invention further includes pharmaceutical compositions containing these compounds and methods of using the same.
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Total number of triples: 506.