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publicationDate 2008-11-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2008293770-A1
titleOfInvention Compounds Which Have Activity at M1 Receptor and Their Uses In Medicine
abstract Compounds of formula (I) and salts are provided: n n n n n n n n n n wherein R 5 is selected from halogen, C 1-6 alkyl, C 1-6 alkyl substituted with one or more fluorine atoms, C 1-6 alkoxy, C 1-6 alkoxy substituted with one or more fluorine atoms, and cyano; R 6 is selected from halogen, C 1-6 alkyl, C 1-6 alkyl substituted with one or more fluorine atoms, C 3-6 cycloalkyl, C 3-6 cycloalkyl substituted with one or more fluorine atoms, C 1-6 alkoxy, C 1-6 alkoxy substituted with one or more fluorine atoms, and cyano; and Q is hydrogen or C 1-6 alkyl. The compounds are M 1 agonists and are useful for therapy, for example in the treatment of psychotic disorders and cognitive impairment.
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Total number of triples: 2091.