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filingDate 2007-04-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2008-10-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2008269228-A1
titleOfInvention Hydrazide-containing hepatitis c serine protease inhibitors
abstract The present invention relates to novel hydrazide-containing compounds of Formula I or Formula II, including pharmaceutically acceptable salts, esters, or prodrugs thereof which inhibit serine protease activity, particularly the activity of hepatitis C virus (HCV) NS3-NS4A protease. Consequently, the compounds of the present invention interfere with the life cycle of the hepatitis C virus and are also useful as antiviral agents. The present invention further relates to pharmaceutical compositions comprising the aforementioned compounds for administration to a subject suffering from HCV infection. The invention also relates to methods of treating an HCV infection in a subject by administering a pharmaceutical composition comprising the compounds of the present invention.
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Total number of triples: 1204.