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publicationDate 2008-10-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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titleOfInvention Monomethylvaline compounds capable of conjugation to ligands
abstract Auristatin peptides, including MeVal-Val-Dil-Dap-Norephedrine (MMAE) and MeVal-Val-Dil-Dap-Phe (MMAF), were prepared and attached to Ligands through various linkers, including maleimidocaproyl-val-cit-PAB. The resulting ligand drug conjugates were active in vitro and in vivo.
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Total number of triples: 2373.