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filingDate 2006-10-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c4a47a1633c52fea387110eb6de37441
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publicationDate 2008-09-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2008213190-A1
titleOfInvention Selective Alfavbetas Receptor Peptide Antagonist for Therapeutic and Diagnostic Applications
abstract The present invention is related to new peptide antagonists of α v β 3 receptor, designed on the basis of the crystal structure of integrin α v β 3 in complex with c(RGDf[NMe]V) and the NMR structure of echistatin. These peptides are potent and selective antagonists of the α v β 3 receptor and can be used as novel anticancer drugs and/or new class of diagnostic non-invasive tracers as suitable tools for α v β 3 -targeted therapy and imaging.
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priorityDate 2005-10-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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