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publicationDate 2008-08-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2008194629-A1
titleOfInvention 3-Mono-and 3,5-Disubstituted Piperidine Derivatives as Renin Inhibitors
abstract The invention relates to 3,5-piperidine compounds, these compounds for use in the diagnostic and therapeutic treatment of a warm-blooded animal, especially for the treatment of a disease (=disorder) that depends on activity of renin; the use of a compound of that class for the preparation of a pharmaceutical formulation for the treatment of a disease that depends on activity of renin; the use of a compound of that class in the treatment of a disease that depends on activity of renin; pharmaceutical formulations comprising a 3,5-piperidine compound, and/or a method of treatment comprising administering a 3,5-piperidine compound, a method for the manufacture of a 3,5-piperidine compound, and novel intermediates and partial steps for their synthesis. Especially, the 3,5-piperidine compounds have the formula I, wherein the symbols have the meanings described in the specification.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410005437
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID142291221
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21829041
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22169820
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129826180
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69137183
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422200153
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID245109744
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID247624120
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID78339
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18521
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID76688
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69137182
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414025133
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID247613193
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID142398595
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID142661138
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID224199348
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226435026
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID224199350
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128585352
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID224199349

Total number of triples: 4097.