http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2008182288-A1

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filingDate 2008-03-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2008-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2008182288-A1
titleOfInvention High-Throughput Screen For Identifying Selective Persistent Sodium Channels Channel Blockers
abstract A method for identifying a selective persistent Na + channel blocker by measuring the ability of the blocker to reduce or inhibit a persistent Na + current to a greater degree than a transient Na + current. Aspects of the present method provide Na + depletion/repletion methods for identifying a selective blocker of a persistent Na + channel, hyperpolarization methods for identifying a blocker of a persistent Na + channel, and Na/K ATPase pump inhibitor methods for identifying a selective blocker of a persistent Na + channel.
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Total number of triples: 604.