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filingDate 2006-03-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_73225eba8d9c3d34aa0bec0339cfd14b
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publicationDate 2007-09-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2007224115-A1
titleOfInvention Polymeric chelators for radionuclide delivery systems
abstract A radionuclide delivery system that is based upon amorphous, water-soluble polymeric chelators. Each water-soluble polymeric chelator is capable of delivering hundreds of radionuclide atoms to the target. The chemical and physical characteristics of the globular polymer increase the effective decay-particle yield at the target cells and reduce ancillary toxicity due to errant daughter radionuclides by retaining or rebinding daughter nuclei. The delivery system includes a water-soluble polymeric chelator having a plurality of chelating groups; and a plurality of radionuclide atoms bound to a least a portion of the chelating groups, wherein the plurality of chelating groups immobilize at least a portion of the plurality of radionuclide atoms.
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